Kev Txhaj Tshuaj-HydroxyPropyl Beta Cyclododextrin
HydroxyPropyl -Clodextrin yog ib qho ntawm cyclodextrin derivatives uas tau kawm ntau yam thiab thov feem ntau ntawm tam sim no. (Rau kev txhaj tshuaj) hydroxypropyl -chlodextrin yog dawb amorphous lossis crystalline ultrafle particle tsis muaj ntxhiab tsw thiab nrog lub qab zib me ntsis. Nws yog ib qho zoo tshaj plaws stubilizer rau kev txhaj tshuaj thiab tshuaj khaws cia.
Cov Lus Qhia Yooj Yim
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Khoom npe |
Kws Tshuaj-qib HYroxyPropyl Beta-Cyclodextrin |
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Cov Qauv Qauv Zoo |
USP-NF 2023 |
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Tsos thiab duab |
Cov hmoov dawb lossis cov khoom siv ultrafine |
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Cas Tsis tau. |
128446-35-5 |
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Molecular Cov Qauv |
C42H70-Tsis35(C3H7O)n |
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Molecular hnyav |
1134.98 + 58n |
Cov Qauv Qauv Zoo
| Kev Txhaj Tshuaj-HydroxyPropyl Beta Cyclododextrin | |||
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Tshuaj Ntsuam Xyuas Tus Qauv |
CHP2020 |
USP-NF2024 |
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Kuaj cov khoom |
Cov Qauv Kev Lag Luam |
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Cov Khoom Siv |
Cov khoom no yog xim dawb lossis tawv dawb los yog cov hmoov uas muaj crystalline, tsw ntxhiab, qab zib, thiab hygroscopic zoo nkauj. Nws yog soluble nyob rau hauv dej, yooj yim soluble hauv ethanol, thiab yuav luag Insoluble hauv acetone. |
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pH |
5.0-8.5 |
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Tshuaj Clarity thiab Xim |
Yuav tsum muaj meej thiab tsis muaj xim |
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Raug Rho Tawm Suab |
Kev nqus tau nyob rau hauv lub wavelength ntau ntawm {0}}}}} nm yuav tsum tsis pub tshaj 0.5 Kev nqus tau nyob rau hauv lub wavelength ntau ntawm {0}}}}} nm yuav tsum tsis pub tshaj 0.5 |
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Kev coj ua |
Tsawg dua los yog sib luag rau 200μs \/ cm |
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Tshuaj ntsuab |
Tsawg dua li lossis sib npaug rau 0. 05% |
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Hydroxyprropoxy cov ntsiab lus |
17.5%-29.1% |
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Dej Cov Ntsiab Lus |
Tsawg dua los yog sib npaug rau 6. 0% |
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Lwm yam tshuaj |
Gamma cyclodextrin |
Tsawg dua los yog sib npaug rau 1.5% |
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1, {2-} propylene glycol |
Tsawg dua los yog sib npaug rau 0. 5% |
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Lwm yam tsis txaus ntseeg (tshwj tsis yog GAMMA Cyclodextrin thiab 1, 2-}} ecylene glycol) |
Tsawg dua los yog sib npaug rau 0. 1% |
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Tag nrho ntawm lwm cov impurities (tshwj tsis yog gamla cyclodextrin thiab 1, 2-} ecylene glycol) |
Tsawg dua los yog sib npaug rau 1. 0% |
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Residue ntawm ignition |
Tsawg dua los yog sib npaug rau 0. 2% |
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Cov hlau hnyav |
Tsawg dua los yog sib npaug rau 10ppm |
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Propylene Oxide |
Tsawg dua los yog sib npaug rau 1ppm |
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Microbial txwv |
Tag nrho cov kab mob aerobic |
Tsawg dua li lossis sib npaug rau 1000cfu \/ g |
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Tag nrho cov pwm thiab cov poov xab suav |
Tsawg dua los yog sib npaug rau 100cfu \/ g |
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Escherichia coli |
Tsis kuaj tau |
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Tus ntses siav |
Tsis kuaj tau |
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Bacterial endotoxins |
Raws li cov kev xav tau |
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Cov khoom lag luam
Kev qhia txog ntawm hydroxyprropyl tsoo cov benamolecular hydrogen bonds tsis pub dhau -cychlodextrin thiab ua rau nws txhaj tshuaj zoo tshaj plaws thiab kev zam. Nws cov haujlwm tseem ceeb hauv cov chaw tshuaj yog li hauv qab no:
1. Nce lub solubility ntawm cov tshuaj, uas tuaj yeem txhim kho lub hydrophilicity ntawm tsis zoo soluble thiab roj-soluble tshuaj;
2. Kev tswj hwm lossis tswj cov tshuaj tso tawm, tiv thaiv kev ua yeeb tshuaj ntawm cov tshuaj, thiab muaj cov kev thov kev pab zoo hauv cov tshuaj tiv thaiv tshuaj;
3. Txhim kho cov xyoob tshuaj, ua kom muaj kev npaj tshuaj lossis txo qis npaum li cas.
4. Txo cov tshuaj lom rau cov tshuaj lom los ntawm cov tshuaj, npog ntsej muag tsw tsw qab;
5. Txhim kho cov khoom siv ntawm cov tshuaj, thiab txhim kho kev ruaj khov yeeb tshuaj.
Cov tau txais daim ntawv thov
Injectable grade hydroxypropyl -cyclodextrin can be used in injectable formulations, mucosal delivery systems (including nasal mucosa, rectum, cornea, etc.), transdermal drug delivery systems, carriers for lipophilic targeted drugs, and also can be used as protectants and stabilizers for proteins.
Ntim thiab Ntim Khoom
- NTIM NTAU: 100G \/ 500G \/ 1KG \/ 2KG \/ 10KG
- Daim Ntawv Ntim: Kev Kho Mob Tsawg-Ntawj Polyethylene Hnab + Tag nrho Cov Ntawv Chim Los Yog Cardboard Chim
- Kev Cia Cov Txheej Txheem: Khw hauv qhov chaw tsaus thiab kaw
Cim npe nrov: HydroxyPropyl Beta Cyclododextrin Kev txhaj tshuaj, Tuam Tshoj HydroxyPropyl Beta CyclodExtrin rau Kev Txhaj Tshuaj Rau Kev Txhaj Tshuaj, cov chaw muag khoom, Hoobkas
