Cov kab mob gram-tsis zoo muaj kev tiv thaiv muaj zog tiv thaiv cov tshuaj tua kab mob vim yog qhov thaiv kev sib luag ntawm lawv cov membrane sab nraud. Tsis ntev los no muaj kev tsim qauv ntawm cov tshuaj tshiab, PPA148, uas qhia tau cov haujlwm zoo tawm tsam txhua tus kab mob gram-tsis zoo. Qhov no yog tshaj tawm cov tshuaj tua kab mob kab mob-cyclodextrin-liposome (ACL) cov kab mob Hydrophobic ppa148, uas tau qhia cov kab mob Hydrophobic ppa148, uas qhia cov kab mob Hydrophobic ppa148, uas tau qhia cov kab mob Hydrophobic ppa148, uas tau qhia cov kab mob Hydrophobic ppa148, uas tau qhia cov kab mob Hydrophobic ppa148, uas qhia cov kab mob Hydrophobic ppa148, uas tau qhia cov kab mob Hydrophobic ppa148, uas tau qhia cov kab mob zoo rau cov kab mob tsis zoo.
Aqueous solubility ntawm cov tshuaj tau txhim kho los ntawm kev sib cuam tshuam nrog ob qho hloov kho betaccylodextrin (HPBCD) thiab Methyl Betaclodextrin (rameb). Txawm hais tias tsis muaj qhov sib txawv ntawm cov kab mob ARL ntawm cov kab mob hauv lub hnab ntawv \/ CD txheej txheem ntawm cov qib molecular siv cov txuj ci nruab nrab siv interfacial cov tswv yim. Cov txiaj ntsig qhia hais tias Liposomes ua raws li cov neeg nqa khoom ntawm cov nyom, fusing rau cov tso tawm sab nraud thiab yog li txhawb nqa daim ntawv tso tawm, thaum RameB tseem tuaj yeem thauj los ntawm sab hauv membrane. Neuron Refrown tau ua tiav los ua kom pom lub hnab ntim khoom siv tau thaum muaj kev cuam tshuam nrog tus qauv sab nraud.
Qhov kev kawm no qhia tau tias ACLs cog lus rau hydrophobic vectors, ob qho yeeb tshuaj tshiab thiab cov uas tau ua tsis tiav vim yog vectors 'tsis kam. ACL cov qauv yuav pab tau nyob rau hauv kev tawm tsam amr raws li lawv lub hom phiaj Om thiab txhij ntawm gram-tsis zoo rau cov solubility ntawm cov solubility ntawm cov solubility ntawm cov tshuaj, yog li nce nws cov bioavailability.
